Home
Publishing
DrugRxiv
Drug Repurposing
Network Medicine
About
REPO4EU
Meet the team
Drug Repurposing Research Collection
Conference
Blog
My ScienceOpen
Sign in
Register
Dashboard
Search
Home
Publishing
DrugRxiv
Drug Repurposing
Network Medicine
About
REPO4EU
Meet the team
Drug Repurposing Research Collection
Conference
My ScienceOpen
Sign in
Register
Dashboard
Search
44
views
0
references
Top references
cited by
1
Cite as...
0 reviews
Review
0
comments
Comment
0
recommends
+1
Recommend
0
collections
Add to
0
shares
Share
Twitter
Sina Weibo
Facebook
Email
3,293
similar
All similar
Record
: found
Abstract
: not found
Book
: not found
Peptides: The Wave of the Future
other
Editor(s):
Michal Lebl
,
Richard A. Houghten
Publication date
(Print):
2001
Publisher:
Springer Netherlands
Read this book at
Publisher
Buy book
Review
Review book
Invite someone to review
Bookmark
Cite as...
There is no author summary for this book yet. Authors can add summaries to their books on ScienceOpen to make them more accessible to a non-specialist audience.
Related collections
Future Science Group
Author and book information
Book
ISBN (Print):
978-94-010-3905-5
ISBN (Electronic):
978-94-010-0464-0
Publication date (Print):
2001
DOI:
10.1007/978-94-010-0464-0
SO-VID:
26fe4748-e73d-477a-a79b-581bfea2dee2
History
Data availability:
Comments
Comment on this book
Sign in to comment
Book chapters
pp. 3
From Merrifield to MetaPhore: A Random Walk with Serendipity
pp. 13
Genomics: From Microbes to Man
pp. 17
Fluorous Methods for Synthesis and Separation of Organic Molecules: From Separating Mixtures to Making Mixtures
pp. 20
Synthesis of β and γ-Substituted Prolines for Conformation-Activity Relationship Studies of the α-MSH Analogue MT-II
pp. 22
The General Asymmetric Synthesis of Syn- and Anti-β-substituted Cysteine and Serine Derivatives
pp. 24
The Novel Asymmetric Synthesis of β-Functionalized Phenylalanine Derivatives
pp. 26
An Efficient Method for Large-Scale Synthesis of Stereochemically Defined and Conformationally Constrained β-Substituted or α,β-Disubstituted Amino Acids
pp. 28
Synthesis of Amino Acids with Novel Biophysical Properties
pp. 30
Two Novel and Efficient Approaches to Synthesis of Enantiopure Dipeptide β-Turn Mimetics: Indolizidinone Amino Acids
pp. 32
Enantioselective Synthesis of β2-Homotryptophan for a Somatostatin Mimetic
pp. 34
Ethyl Nitroacetate as a Useful Synthon for the Synthesis of Orthogonally Protected, Poly-Functional Cαα-Disubstituted Amino Acids
pp. 36
Synthesis of β-Benzo[b]thiophene Dehydroamino Acids by Suzuki Palladium Catalyzed Cross Coupling
pp. 38
Efficient Diastereoselective Synthesis of a Hydroxyethylene Dipeptide Isostere
pp. 40
One-Pot Conversion of Azides to Protected Guanidines via the Staudinger Reduction; Synthesis and Utilization of the Phe-Arg Hydroxyethylene Dipeptide Isostere
pp. 42
The Synthesis of Tyrosine Mimetics via a Novel N(1)-C(4) Beta-Lactam Cleavage Reaction
pp. 44
Michael Additions to Dehydroalanine Derivatives
pp. 46
Facile Synthesis of a Constrained Dipeptide Unit (DPU) for Use as a β-Sheet Promoter
pp. 48
Synthesis of N α-(Fluoren-9-ylmethoxycarbonyl)-N ε-[(7- methoxycoumarin-4-yl)-acetyl]-L-lysine for Use in Solid-Phase Synthesis of Fluorogenic Substrates
pp. 50
Preparation of β-Amino-α-mercapto Acids and Amides: Stereocontrolled Syntheses of 2′-Sulfur Analogues of the Taxol C-13 Side Chain, Both syn and and S-Acetyl-N-benzoyl-3-phenylisocysteine
pp. 52
New Approach for Preparation of C-Glycoamino Acid Building Blocks
pp. 54
New Quencher Derivatives for Fluorescence Quenching Peptide Assays
pp. 56
Preparation of (2S)-2-Amino-3-(2-(2,2,5,7,8-pentamethylchroman-6-sulfonyl)-1H-indol-3-yl)-propionic acid and Its Incorporation into Antibacterial Lactoferricin Peptides
pp. 58
UniChemo Protection (UCP)
pp. 61
An Improved Synthesis of Fmoc-Asp(O-3-methylpent-3-yl)-OH, an Aspartate Derivative That Resists Base Induced Aspartimide Formation
pp. 63
Systematic Investigation of the Aspartimide Problem
pp. 65
Ninhydrin as a Reversible Protecting Group of N-Terminal Cysteine
pp. 67
Novel Synthesis and Application of a Protected Bicyclic α-Helix-Initiating Heptapeptide Suitable for Segment Condensation Syntheses: Utility of Pentaaminecobalt(III) for Carboxyl Protection
pp. 69
Nin-4-Nitrobenzenesulfonyl Tryptophan: A Convenient Preparation of N α-Boc and N α-Fmoc Derivatives
pp. 71
Syntheses of Difficult Hydrophobic Sequences Using 2-(4-Nitrophenyl)sulfonylethoxycarbonyl(Nsc)-N α-(2-hydroxy- 4-methoxybenzyl)Ala-OH: (Ala)10-Valine, (Ala)15-Valine
pp. 73
A Highly Efficient Method for Synthesis of Fmoc-Lysine(Mmt)-OH
pp. 75
A New Practical Approach to the Synthesis of Fmoc-L-Cysteine
pp. 77
A Novel Protocol of Solid Phase Peptide Synthesis with 2-(4-Nitrophenyl)sulfonylethoxycarbonyl(Nsc)-Amino Acids
pp. 79
S-Xanthenyl Protected 1-Thiosugars as Building Blocks for Glycopeptide Assembly
pp. 81
Late Deprotection Difficulties During SPPS Depend on the Preceding Sequence
pp. 83
Towards a Selective Boc Deprotection on Acid Cleavable Resin
pp. 85
By-Product Formation During SPPS of Linear, Cyclic, and Novel Bicyclic Peptides as AChE Inhibitors
pp. 87
Acidic Cleavage of the Side Chain Protecting Groups of Peptides Attached to a Modified Polystyrene Carrier: Synthesis of Peptide Generics
pp. 89
The Use of a Novel Safety Catch Linker for BOC-Based Assembly of Cyclic Peptide Libraries
pp. 91
Diurethanyl 1H-Benzotriazole-1-carboxamidines as Guanidinylating Reagents
pp. 93
Amino Acid Bromides: A Convenient Choice for Very Difficult Couplings
pp. 95
Synthesis of the Two Isomeric Benzo Derivatives of 1-Hydroxy-7-azabenzotriazole and Preliminary Studies of Their Effectiveness as Coupling Reagents
pp. 97
Optimization of Coupling Methods for the Introduction of Mono-Benzyl Phosphate Esters of Fmoc Protected Phosphoamino Acids
pp. 99
HATU-HOAt-CuCl2: A Reliable Racemization-Free Segment Coupling System
pp. 101
Search for a Safe, Inexpensive and Convenient Amidation Process for Protected Amino Acids and/or Peptides
pp. 103
Extending Synthetic Access to Proteins
pp. 105
A New Scaffold for Amide Ligation
pp. 107
Chemical Ligation of Multiple Peptide Fragments Using a New Protection Strategy
pp. 109
Synthesis of Oligodeoxynucleotide-Peptide Conjugates Using Hydrazone Chemical Ligation
pp. 111
The Use of a Free Peptide for Preparation of a C-Terminal Building Block for Polypeptide Synthesis in Combination with a Peptide Thioester
pp. 113
Synthesis of N to C Terminal Cyclic Analogues of α-Conotoxin Iml by Chemoselective Ligation of Unprotected Linear Precursors
pp. 115
Total Chemical Synthesis of κ-Casein Using Native Ligation Methodology
pp. 117
Fmoc Chemistry Compatible Methods for Thio-Ligation Assembly of Proteins
pp. 119
Simultaneous Lipidation of a Multi-Epitope Peptide Cocktail by Chemoselective Hydrazone Formation
pp. 122
Privilege Structures: New Strategies for the Synthesis of Cyclic Tetrapeptides
pp. 125
Incorporation of a cis-Amide Bond Isostere in the Synthesis of Cyclic Tetrapeptides
pp. 127
Covalent Control of Shape and Folding in Peptides by Ring-Closing Metathesis
pp. 130
New Synthetic Routes to NEtXaa4-Cyclosporin Derivatives as Potential Anti-HIV Drugs
pp. 132
Transition Metal Complexes of Linear and Cyclic Pseudopeptides
pp. 134
An Efficient Synthesis of Integrin Antagonists cyclo(-RGDfK-), cyclo(-GRGDfK-) and Their Conjugates with MAG3 Chelate
pp. 136
Design and Synthesis of Cyclic Peptide Antagonists Intended to Block Coactivator Binding to Steroid Nuclear Receptors
pp. 138
A Novel Design and Synthesis of Bicyclic Peptide Library
pp. 140
Strategies for the Synthesis of Cyclic Peptides
pp. 142
Vinyl Sulfide Cyclized Analogues of Angiotensin II with High Affinity to the AT1-Receptor
pp. 144
Strategies for the Synthesis of Novel Head-to-Side Chain Cyclic Peptides: Application to Dynorphin A Analogs
pp. 146
Study on the Influence of Different Metal Ions on Cyclization of Linear Pentapeptides and Heptapeptide
pp. 148
Disulfide Bond Formation of a Hydrophobic Peptide by Dimethyl Sulfoxide
pp. 150
Stereoselective Synthesis of Transition State Analog Inhibitors of DPP-IV Using 2-Substituted Thiazoles
pp. 152
Original and General Strategy of Dimerization of Bioactive Molecules
pp. 155
An Efficient Approach for the Synthesis of Salmon Calcitonin Using Oxazolidine Dipeptides
pp. 157
A Combined Solid-Phase and Solution Strategy for Chemical Synthesis of Human Leptin
pp. 160
Synthesis of Phosphorylated Polypeptide by the Thioester Method Using a Recombinant Protein
pp. 162
The Synthesis of the K-Ras-Derived Peptide
pp. 164
Synthesis of Phosphopeptides on Solid Phase Using tert-Butyl-H-phosphonate Salts
pp. 166
Solid Phase Synthesis of Seleno-Methionine Peptides by tBoc/Bzl and Fmoc/tBu Protection Strategy Suitable for the Crystallographic Phase Determination by Multi-Wavelength Anomalous Diffraction (MAD)
pp. 168
Synthesis of a C-Terminal Fluorescein-Labeled 36-mer Peptide
pp. 170
Expanding Diversity: Modification of Linear and Cyclic Peptides by C-Glycosylation and N-Methylation
pp. 172
One-Dimensional Spatial Encoding: Split/Mix Synthetic Parallelism with Tag-Free Identification and Assays at the Speed of Light
pp. 174
Spatial Screening of Lectin Ligands. Cyclic Peptides as Scaffolds for Multivalent Presentation of Carbohydrates
pp. 177
Combinatorial Syntheses of Polyhydroxamate Siderophores: Desferrioxamine, Exochelin, Mycobactin, and Aerobactin Libraries
pp. 180
Identification of Peptide Ligands for α4β1 Integrin Receptor as Potential Targeting Agents for Non-Hodgkin’s Lymphoma
pp. 183
Development of Peptidomimetic Substrates and Inhibitors that Bind to the Peptide Binding Pocket of the Catalytic Site of p60c-src Protein Tyrosine Kinase
pp. 185
Pseudoproline Libraries for Tuning Inhibitors of SH3 Domain Mediated Protein-Protein Interactions
pp. 187
Towards a Set of Peptides with Orthogonal HIV Seroreactivity Using Adaptively Coded Peptide Libraries: Decoding by Mass Spectrometry and Immunofluorescent Screening
pp. 189
Mapping of Discontinuous Epitopes on FSH
pp. 191
Development of Highly Specific, Membrane Permeable Peptide Blockers of cGMP-Dependent Protein Kinase Utilizing Affinity Selection from Peptide Libraries
pp. 194
The Integration of Positional Scanning Libraries with Bioinformatics and Proteomics
pp. 196
Screening and Synthesis of a Positional Scanning Library Based on the Bowman-Birk Reactive Site Loop
pp. 198
A Bicyclic Peptide Template Useful for Solution-Phase Combinatorial Synthesis
pp. 200
Synthesis of Combinatorial Libraries Associated with Constrained β-Turn Mimetics
pp. 202
Screening and Design of Hybrid Peptide That Binds with Glucose Oxidase
pp. 204
Combinatorial Synthesis, Screening and Testing of Peptidic RNA-Ligands
pp. 206
High Throughput Peptide Syntheses Generate Ligands for Proteomic Database
pp. 208
MHC Ligand Motifs from Peptide Libraries: The Software EPIPREDICT
pp. 210
High-Density Compound Arrays of Combinatorial Chemical Libraries by a New Pen-Directed and Computer-Navigated Plotter Device
pp. 212
Combining SPOT Synthesis and Native Chemical Ligation to Generate Large Arrays of Small Protein Domains
pp. 214
Peptides as Drugs: Is There a Market?
pp. 217
Solid-Phase Total Syntheses of Trunkamide A and Kahalalide F, Cyclic Peptides from Marine Origin
pp. 220
Solid Phase Synthesis of Large Cyclic Peptides
pp. 222
Solid-Phase Synthesis of Consolidated Ligands Containing an Intramolecular Lactam Bridge: Comparison of Strategies and Tactics
pp. 224
Backbone Amide Linker (BAL)/Fmoc Synthesis of Peptide Thioester Intermediates Required for Native Chemical Ligation
pp. 226
Ampullosporin Analogs: Solid Phase Synthesis, Conformational Studies, and Biological Activities
pp. 228
Synthesis of Lanthionine-Containing Peptides on Solid Phase via an Orthogonal Protecting Group Strategy
pp. 230
Systematic Solid Phase Synthesis of Linear Pseudooligolysines Containing Multiple Adjacent CH2NH Amide Bond Surrogates: Potential Agents for Gene Delivery
pp. 232
Peptide Transformation and Synthesis of Oligopeptidomimetics
pp. 234
A New Strategy for Inverse Solid-Phase Peptide Synthesis
pp. 236
Optimization of the Chemical Synthesis of Human Ghrelin
pp. 238
Rational Design and Synthesis of a Potent Amide-Linked Cyclic Analogue of MBP87–99 Based on 2D-NMR Studies and Molecular Dynamics
pp. 240
Solid-Phase Synthesis Utilizing Azido-α-Amino Acids: Reduction of Azido-Protected Proline
pp. 242
Improved Fmoc-Solid Phase Synthesis of β-Amyloid Peptides Using DBU as Nα-Deprotection Reagent
pp. 244
Triphosgene as Peptide Coupling Reagent: Highly Efficient Total Synthesis of Cyclosporin O
pp. 246
Synthesis of Ferrocene Linkers for Solid-Phase Synthesis of Peptides
pp. 248
Efficient HF Conditions for Suppressing Trp Modification Associated with Use of the N in-Cyclohexyloxycarbonyl (Hoc) Group
pp. 250
Structural Characterization of a Dibenzylated-CGRP(8–37), a Byproduct from N-α-Benzylation of CGRP(8–37)
pp. 252
Polyamines as Intermediates for the Synthesis of Heterocyclic Compounds and Oligomeric Heterocyclic Compounds from Resin-Bound Polyamides
pp. 255
Solid-Phase Synthesis of Substituted Dihydroimidazoles and Their Bis Analogs
pp. 257
Solid Phase Synthesis of 1,2,5-Substituted Derivatives of 4-Imidazolidinone
pp. 259
Solid Phase Synthesis of 1,2,4-Triazinan-3-ones
pp. 261
Solid-Phase Synthesis of α-Difluoro-β-amino Acids by a Reformatsky Reaction
pp. 263
Peptidotriazoles: Copper(I)-Catalyzed 1,3-Dipolar Cycloadditions on Solid-Phase
pp. 265
Solid-Phase Synthesis of Lidocaine Analogues Using Backbone Amide Linker (BAL) Anchoring
pp. 267
Solid-Supported Triazenes as Alkylating Polymers Employed for the Versatile Derivatization of Peptides
pp. 269
Oxidation of Threonine and Serine Residues on Solid-Phase: Pyrazine Formation by Dess-Martin Periodinane Oxidation
pp. 271
A Novel Solid Phase Approach to Thioether Cyclized Peptides: Discovery of Mouse Melanocortin-1 Receptor Agonists
pp. 273
Bifurcated Dipeptide Schiff Bases as Ligands for Enantioselective Catalysis: Micro-Metalloenzymes
pp. 275
Recent Advances in the Solid-Phase Synthesis of Long-Chain β-Peptides
pp. 277
Fully Automated Parallel Oligonucleotide Synthesizer
pp. 279
N to C Solid Phase Organic Synthesis of Peptidic and Peptidomimetic Derivatives Using 9-Fluorenylmethyl Esters
pp. 283
A New Method to Quantify the Swelling Properties of Polymer Beads Used in Solid Phase Peptide Synthesis (SPPS)
pp. 285
A Novel High Throughput Analysis of Total Nitrogen Content by a Colorimetric Method
pp. 287
Conformational Studies of Cyclotetrapeptides [Xaa-D-Ala]2 by NMR, CD and Molecular Modeling
pp. 289
Conformation of β3-Residues-Containing Cyclic Pentapeptide Analogues of the Antitumoral Astin Family
pp. 291
Structure-Activity Relationship of Antimicrobial Peptide, Gaegurin 4, Isolated from Korean Frog
pp. 293
Tethering of the Proximal Region of the Angiotensin II Receptor (AT1A) C-Terminus to the Cell Membrane
pp. 295
Amide I Frequency as a Probe of Tertiary Structure: FTIR Studies of Helix Bundle Peptides
pp. 297
Coupled Plasmon Waveguide Resonance Studies of Agonist/Antagonist Binding to the Human δ-Opioid Receptor Provide New Structural Insights Into the Three-State Model for Receptor-Ligand Interactions
pp. 299
Structure Elucidation of Peptides with Unnatural Amino Acids Using an Automated Protein Sequencer
pp. 301
Structural Study of the Pro-Sequence of Protegrin-3
pp. 303
α-Helix Stabilizing Aromatic-Backbone Interactions
pp. 306
Solution Structure of Oligopeptides-Copper(II) Complexes
pp. 308
Development of Antibodies Against Conjugated Benzophenone, as a Tool in Photoaffinity Crosslinking Studies
pp. 310
Monitoring Peptide-Induced Liposome Breakdown with Fluorescence Correlation Spectroscopy
pp. 312
NMR Structural Investigation of a β3-Dodecapeptide with Proteinogenic Side Chains in MeOH and Water
pp. 314
Conformational Studies on a Synthetic Peptide with Prolactin-Releasing Activity in a Membrane Mimetic Environment
pp. 316
Analysis and Characterization of Combinatorial Mixtures of Mucin-2 Antigen Peptides
pp. 318
High Throughput Validation and Quantitation of Synthetic Peptides via LC-MS
pp. 320
Synthesis and Solution Three-Dimensional Structure of the Immunodominant Region of Protein G of Human RSV
pp. 322
Role of Residues in Position 2 and 7 on the Conformation of the N-Terminal Apamin Loop
pp. 324
Conformational Study of [desHis1, desPhe6, Glu9]glucagon-NH2 by 2D-NMR Spectroscopy in the Presence of Perdeuterated Dodecylphosphocholine
pp. 326
Molecular Modeling Study of the β-Turn-Type Reversals Involved in 3D Structure of IFABP
pp. 328
Structural Features of Short, Linear Peptides in Solution by Fluorescence and Molecular Mechanics Studies
pp. 330
Influence of Stereochemistry of the Preceding Acyl Residue on the cis/trans Ratio of the Proline Peptide Bond
pp. 332
The Influence of the Surrounding Media on the Structural Propensities of Amino Acid Residues in Proteins
pp. 334
CD Evidence of the Conformational Transitions in rMOG[1–125] in the Presence of Membrane Mimicking Detergents
pp. 336
Coacervation and CD and FT-IR Spectroscopic Studies of Elastin-Derived Polypentapeptide and Its Analogs
pp. 338
Conformational Analysis of Human Calcitonin in Aqueous Solution and Comparison with a Highly Potent Lactam-Bridged Analogue
pp. 340
Conformational Studies of a Glycopeptide Recognized with High Affinity by Autoantibodies in Multiple Sclerosis
pp. 342
Human Relaxin Chain Combination and Folding
pp. 344
Effects of Human Leptin Fragments in Hypothalamic Nucleus C-Fos Expression
pp. 346
Introduction of Temperature-Sensitive Elastin-Based Switches to Stabilize Globular Proteins
pp. 348
A Short-Range Interaction of the cis-trans Urea Motif in Ureapeptides
pp. 350
A New N-Terminal Helix Capping Box
pp. 353
The Determination of Helix Stability Coefficients Using D-Amino Acid Substitutions in the non-Polar Face of an Amphipathic α-Helical Model Peptide
pp. 355
NMR-Based Studies of a Collagenous Substrate of Collagenase
pp. 357
Conformational Analysis of Model Polypeptides Having Repetitive Xaa-Pro Sequences
pp. 359
The Role of Unstructured Highly Charged Regions on the Stability and Specificity of Dimerization of Two-Stranded α-Helical Coiled-Coils: Neck Region of Kinesin-Like Motor Protein Kif3A
pp. 361
A Leu-Thr-Trp-Lys “Lock” Stabilizes the N-Terminus of the Kinesin Neck Coiled-Coil
pp. 363
Template-Assisted Stabilization of a Short HIV-1 gp41 Inner-Core Coiled-Coil Peptide
pp. 365
STABLECOIL: An Algorithm Designed to Predict the Location and Relative Stability of Coiled-Coils in Native Protein Sequences
pp. 367
Stabilization of Helical Conformation in Model Peptides by 2,2,2-Trifluoroethanol: An FTIR Study
pp. 369
Peptides Based on Daf, the First Rigid, Transition-Metal Receptor: Cα,α-Disubstituted Glycine
pp. 371
Allyl-Based, Cα-Methylated α-Amino Acids in the Side-Chain to Side-Chain Ring-Closing Metathesis Reaction of β-Turn/310-Helical Peptides
pp. 373
Synthesis and Conformational Analysis of Polypeptides Having Repetitive Xaa-Pro-Pro Sequences
pp. 375
Biophysical Studies of a Proline-Rich Peptide from the Coral Bleach Pathogen Vibrio shiloi
pp. 377
Lactam-Bridged and Disulfide-Bridged Peptide Mimic of a Stable α-Helical Folded Protein
pp. 379
Stabilization of the Triple Helix of Collagen Peptides Using Fluoroproline and/or Triacid Scaffolds
pp. 381
Conformational Studies of O-Glycosylated 15-Residue Peptide from the Human Mucin (MUC1) Protein Core
pp. 383
Folding of β- and γ-Peptides — the Influence of Substitution Patterns on the Formation of Secondary Structures
pp. 385
The β-Methyne of Ile3 in the Propeptide Region of Prouroguanylin is Crucial for Chaperone Function in the Folding of the Mature Peptide, Uroguanylin
pp. 387
Solution Structure of the Macrocyclic Squash Trypsin Inhibitor MCoTI-II, the First Member of a New Family of Cyclic Knottins
pp. 389
Delineation of Structural Constraints Imposed by a Dimerizer Peptide When Grafted Onto the Terminal Ends of a Test Peptide
pp. 391
Local and Long-Range Sequence Contributions to the Folding of a Predominantly β-Sheet Protein
pp. 394
3D Models for Conformational States of the V3 and V1/V2 Loops in gpl20/CD4/Antibody Complex
pp. 396
Structure and Dynamics of Ribosome Recycling Factor
pp. 398
Peptide Models for Studying Autonomous Folding of Subdomain Sections of Protein Molecules
pp. 400
Towards New Designed Proteins: Oxime Ligation of Core Modules
pp. 402
Do Bioactive Peptides Display Native-Like Conformations When Bound to a Solid Support?
pp. 404
Direct Observation of Backbone Hydrogen Bonding in the Folding Transition of Chymotrypsin Inhibitor 2 (CI2)
pp. 406
Optimizing Aqueous Fold Stability for Short Polypeptides: 20 Residue Miniprotein Constructs That Melt as High as at 61 °C
pp. 409
Synthetic Approach to Study the Effects of β-Turn Residues on the Structure and Folding of Bovine Pancreatic Trypsin Inhibitor (BPTI)
pp. 411
NMR Solution Structure of B-Motif, a Signature Motif of Type-B Response Regulators for His-to-Asp Phosphorelay Signal Transduction System, and Its Interactions with DNA
pp. 413
Synthesis and Characterization of the Pain-Killing Peptide Grammostola spatulata Analgesic Factor (GsAF-1) Containing Three Disulfide Bonds
pp. 415
Molecular Modeling: Indispensable Tool at the Interface Between Structural Analysis and Molecular Design
pp. 418
Molecular Modeling and Binding Energy Calculations for Drug Resistant Mutations in HIV-1 Protease-Inhibitor Complexes
pp. 420
Electrostatic and Hydrophobic Nature of the Binding of Gelsolin 135–142 and Gelsolin 150–169 Fragments to the PIP2-Containing Lipid Bilayer
pp. 422
Prediction of Antibody Complexes with Rationally-Designed and Library-Derived Cyclic Peptides: A Computer Modeling Study
pp. 424
Ligand-Receptor Interactions Regulating Cell Trafficking and Signaling of the Human PTH1Rc: An in Silica Examination
pp. 426
Theoretical Design of α-Hairpin Structures
pp. 428
Application of a Detailed Energy Surface to Homology Modeling of the ω-Conotoxin Family
pp. 430
DARWINIZER® — a Computer Based Method for Peptide and Peptidomimetics Design
pp. 432
Proline: A Key Building Block in “de novo” Designed Peptide Molecules
pp. 435
Complementary Assembly of Heterogeneous Multiple Peptides into Amyloid Fibrils with α-β Structural Transitions
pp. 438
Conformational Uniqueness via Designed Ion Pairs
pp. 440
Design, Synthesis and Incorporation in Peptides of a β-Turn Mimetic
pp. 442
Evaluating PERMs as Protein Mimics
pp. 444
Amphipathic Stabilization of the 310-/α-Helix Equilibrium in Synthetic Peptides Rich in Cα, Cα-Disubstituted Glycines
pp. 446
Design, Synthesis and Characterization of Novel Scaffold-Assembled Collagen Mimetics
pp. 448
Design and Synthesis of a Mini-Prorelaxin Model
pp. 450
Site Specificity Metal Binding Affinity in C-Terminal of Calmodulin
pp. 452
A Cassette Ribonuclease: Site Selective Cleavage of RNA by a Ribonuclease S-Bearing RNA-Recognition Segment
pp. 454
Protein Models on Carbohydrate Templates: Effect of the Template
pp. 456
New Foldamers: Rigid Peptides with an Alternating cis-trans Amide Sequence
pp. 458
Design, Synthesis, and Conformational Studies of Short Peptides Containing C αα-Dipropylglycine and Dibenzylglycine
pp. 460
Bromo Tryptophan Based Antisickling Peptides: Design, Synthesis and Evaluation
pp. 462
Synthesis, Redox and Structural Properties of Cystine-Cyclopeptides Containing the Active-Site of the Thioredoxin Superfamily
pp. 464
Probing Backbone Flexibility Within the Active Site of Glutaredoxin 3
pp. 466
Homostranded and Heterostranded α-Helical Templates for Combinatorial Library Display: Differences in Stability and Solubility
pp. 468
Synthesis and Solution Structures of Cyclic Hexapeptides Cyclo(Pro-Leu-Xxx)2
pp. 470
Functional and Structural Comparisons of Linear and Dendritic Arrays of Polypeptides
pp. 475
Synthetic Studies on the Antimicrobial Activity of Pleurocidin
pp. 477
Disruption of the β-Sheet Structure of Cyclic Peptides by Single Amino Acid Substitution: Influence on Prokaryotic and Eukaryotic Cell Viability
pp. 479
Relationship Between Amphipathic Secondary Structure and Activity in Model Linear Cationic Antimicrobial Peptides
pp. 481
Shedding Light on the Aglycon Formation of Glycopeptide Antibiotics
pp. 483
Synthesis of λ-Conotoxins, a New Family of Conotoxins with Unique Disulfide Pattern
pp. 485
Solution Conformation of an α-Conotoxin GI with a D-Tyr at Position 11
pp. 487
Antimicrobial and Chemotactic Activities of ω-Conotoxin Cyclic Analogues
pp. 489
Synthesis of Parallel and Antiparallel Magainin 2 Dimers and Their Interaction with Lipid and Cell Membrane
pp. 491
Interaction of the Antimicrobial Peptide PGLa and Its Ala-Substitution Analog with Membrane-Mimetic Systems
pp. 493
Antibacterial Activity Spectrum of Designed Pyrrhocoricin Analogs
pp. 495
Importance of the Intramolecular Disulfide Bridges in the Biological Activity of Gomesin
pp. 497
Variation in Ring Size of Cyclic Antimicrobial Peptides Results in Diversity and Selectivity of Biological Activity
pp. 499
α-Helical Glycopeptide Analgesics: β-Endorphin Mimics with Good in vivo Potency
pp. 502
Efforts to Investigate the Conformational Changes of the Prion Protein by N-Glycosylation
pp. 504
Glycation of Leucine-Enkephalin: Imidazolidinones and Amadori Compounds
pp. 506
Solid-Phase Synthesis of Thio-Linked C-Terminal Glycopeptides via a Mitsunobu Reaction
pp. 508
Synthesis of the Extracellular Ig Domain I (34–94) of Emmprin Carrying a Chitobiose Unit
pp. 510
Synthesis of Peptide- and Glycopeptide-Conjugates for Specific Drug Targeting
pp. 512
Complexation of Peptidoglycan Intermediates by the Lipoglycodepsipeptide Antibiotic Ramoplanin: Structural Requirements for Intermolecular Complexation and Fibril Formation
pp. 514
Short Analogues of the Lipopeptaibol Trichogin GA IV
pp. 516
Dinuclear Zinc(II) Complexes of Linear and Cyclic Peptides Containing Two Bis(2-pyridylmethyl)amino Groups as Catalysts for Hydrolysis of RNA Model Substrate
pp. 518
Construction of RNA-Binding Proteins Having Nucleobase Amino Acids Based on HIV-1 Nucleocapsid Protein
pp. 520
Screening of Peptides that Control Interaction Between Nucleobases from Peptide Libraries Based on Loop Structures
pp. 522
Preparation of a Site-Specifically Labeled Fluorescent Chemokine by Chemical Synthesis
pp. 524
Synthesis, Characterization, and Calorimetric Studies of a Series of Novel Bioconjugates for Selective Targeting of Microbubbles to GPIIbIIIa Receptors on Vascular Thrombi
pp. 526
Energy and Electron Transfer Systems Built in Dendritic Poly(L-lysine)s
pp. 528
Design of Analogs of Trapoxin, Cyl-1, and Chlamydocin for MHC Class-I Molecule Up-Regulation
pp. 530
Backbone Assignment of Gyrase-B P24 Fragment and Its Interactions with the Inhibitor GR122222
pp. 532
Synthetic Progress Towards a TMC-95 Analogue as a Potential Proteasome Inhibitor
pp. 534
Prime Site Binding Inhibitors of the Hepatitis C Virus NS3/4A Serine Protease
pp. 537
Solution and Solid Phase Synthesis of Non-Peptide Peptidomimetic Aspartic Peptidase Inhibitors
pp. 539
Design and Synthesis of Novel Matrix Metalloproteinase Inhibitors
pp. 541
A Novel Continuous Assay for the Mechanistic Characterization of Histone Deacetylases and Homologues Using a Small Molecule Fluorescent Substrate
pp. 543
Peptide Inhibitors of α-Amylase Based on Tendamistat: Synthesis and Kinetic Studies
pp. 545
Structural Studies of the Complex Between Decapeptide Inhibitors and the Serine Protease NS3/4A of Hepatitis C Virus
pp. 547
Synthesis and Activity of a Small Cyclic Protease Inhibitor from Sunflower Seeds, SFTI-1
pp. 549
Different Types of P1 Residues in Peptide-Based Inhibitors of Hepatitis C Virus Full-Length NS3 Protease
pp. 551
Development and Characterization of Potent Peptide Inhibitors of p60c-src PTK Using Pseudosubstrate-Based Inhibitor Design Approach
pp. 553
Use of β-Amino Acids in the Design of Substrate-Based Peptidase Inhibitors
pp. 555
Bivalent Inhibition of Human β-Tryptase: Probing the Distance Between Neighbouring Subunits by Dibasic Inhibitors
pp. 558
A Highly Selective Cell Permeable Peptide Inhibitor of Proprotein Convertase 1: Design, Synthesis and Biological Evaluation in Cellular PC1-Mediated Proteolysis
pp. 561
Bicyclic Peptide Inhibitors of an Epithelial Cell-Derived Transmembrane Protease, Matriptase
pp. 563
Probing the Substrate Specificity of Hepatitis C Virus Nonstructural 3 Protein Serine Protease by Intramolecularly Quenched Fluorogenic Peptide Substrates
pp. 565
Characterization of the Staphylococcus aureus Sortase Transpeptidase: A Novel Target for the Development of Chemotherapeutics Against Gram-Positive Bacteria
pp. 567
Cyclic Octapeptide Inhibitors of the Acetylcholinesterase Peripheral Site: Implications for Inhibition of Nerve Toxins
pp. 569
Homologs of Amino Acids and Explorations into the Worlds of β- and γ-Peptides
pp. 572
Designed Amino Acids That Induce β-Sheet Folding and β-Sheet Interactions in Peptides
pp. 575
Triply-Templated Artificial β-Sheets
pp. 577
Stepwise Peptide-Peptoid Transformation via SPOT Synthesis
pp. 579
SPOT Synthesis of 1,3,5-Trisubstituted Hydantoins on Cellulose Membranes
pp. 581
Synthesis and CD Spectra of β2-(3-Aza-peptides)
pp. 583
Preferred Conformations of Azaamino Acids
pp. 585
Higher Anti-HIV-1 Activity of Peptides Derived from gp41 Carboxyl-Terminal Coiled Coil Structure of HIV-1 89.6 Strain
pp. 587
Synthetic Approach to Dipeptide Mimetics Based on Aminoacyl Incorporation Reaction
pp. 589
Convenient Conversion of Amino Acids to Their N-Hydroxylated Derivatives on a Solid Support: Synthesis of Hydroxamate-Based Pseudo-Peptides
pp. 591
Peptide Bond Modification for Metal Coordination: 1. Metal-Binding Properties of Hydroxamate-Based Pseudo-Peptides
pp. 593
Peptide Bond Modification for Metal Coordination: 2. Metal-Binding Properties of Peptide-Derived Pentaaza-Macrocyclic Templates
pp. 595
Peptide Bond Modification for Metal Coordination: 3. Metal-Binding Properties of Phosphorus-Based Pseudo-peptides
pp. 597
Mimicry of the Backbone and Side-Chain Geometry of Peptide Turns: Synthesis of Novel 4-Substituted Indolizidin-9-one Amino Acids
pp. 599
Employing the Steric Interactions of 5-tert-Butylproline to Control Peptide Folding and Biology
pp. 602
Synthesis of β-Turn Mimetics: [5,5]-Fused Bicyclic γ-Lactam Dipeptide Analogues
pp. 604
Pyridine as a Tripeptidomimetic Scaffold
pp. 606
Synthesis of Fluoroalkene Dipeptide Isosteres Utilizing Organometallic Reagents
pp. 608
Synthesis of Peptide Mimetics and Amino Acid Mimetics Bearing Aminoxy Instead of Amino Group
pp. 610
Design and Synthesis of Amide Isosteres of Phe-Gly: Potential Peptidomimetic Ligands for the Intestinal Oligopeptide Transporter PepT1
pp. 612
β-D-Mannose Based Peptidomimetics in the Design of α4ß1 and α4β7 Antagonists
pp. 614
Design, Synthesis and Modulation of Angiogenesis by Thrombin Receptor Non-Peptide Antagonists
pp. 616
Development of Endomorphin Derivatives with Dual Functions and Studies on Their Three-Dimensional Structure
pp. 618
Stereoselective Synthesis of Tyrψ[CH2O]Phe and Tyrψ[CH2O]Ile, Methylene-oxy Analogs of Oxytocin and [8-Arginine]Vasopressin
pp. 620
Exploration of the DTrp-NMeLys Motif in the Search for Potent Somatostatin Antagonists
pp. 622
Synthesis and Biological Evaluation of Mixed β2/β3-Dipeptides as Somatostatin Analogs
pp. 624
Cyclic Peptides Related to Somatostatin Containing a Novel Imidazole Derived cis-Amide Mimetic
pp. 626
Human Somatostatin Receptor Specificity of Backbone-Cyclic Analogs Containing Novel Sulfur Building Units
pp. 628
Linear and Cyclic Thr6-Bradykinin Analogues Containing N-Benzylglycine as a Replacement for Residues Phe5 and Phe8
pp. 630
Design, Synthesis and Conformational Analysis of Human Urotensin II (U-II) Analogues with Lactam Bridge
pp. 632
PACAP27 Analogues Incorporating Type II/II’ β-Turn Mimetics
pp. 634
Bicyclic β-Strand Templates: Epimerization and Biological Activity of Non-Electrophilic Serine Protease Inhibitors
pp. 636
Design, Synthesis and Biological Evaluation of Pilicides: Inhibitors of Pilus Assembly in Pathogenic Bacteria
pp. 638
Phenylahistin, a Small Dipeptidic Colchicine-Like Anti-Microtubule Agent: Total Synthesis and SAR Study of the Derivatives
pp. 640
New Antiproliferative Agents from a Peptidomimetic Library
pp. 642
Development of New Analogs of the Highly Potent Anti-Cancer Compound BKM-570
pp. 644
Design and Synthesis of a Selective PSA Cleavable Peptide-Doxorubicin Prodrug Which Targets PSA Positive Tumor Cells
pp. 647
Peptidic Inhibitors for Protein-Protein Interactions at Cell Surfaces
pp. 650
Prodrug Forms of Peptidomimetic HIV Protease Inhibitors Using Intramolecular Cyclization Reaction
pp. 652
Effect of Poly[L-Lysine] Based Polymer Polypeptides on Chemotaxis and Phagocytosis of the Unicellular Tetrahymena pyriformis GL
pp. 654
Costimulatory Blockade by CD28 Peptide Mimics: Suppression of Experimental Autoimmune Encephalomyelitis
pp. 656
Design and Synthesis of an Amide-Linked Angiotensin II Analogue with 3,5 Side Chain Bridge: Structural Resemblance of Ring Cluster Conformation with AT1 Non-Peptide Antagonists
pp. 658
Sustained Delivery of an ApolipoproteinE Peptidomimetic Lowers Serum Cholesterol Levels in Dyslipidemic Mice
pp. 660
Design, Synthesis and Biological Evaluation of Novel Non-Peptide Opioid Ligands for Human Pain
pp. 662
Design and Synthesis of Novel Pure Motilin Antagonists
pp. 664
Active Somatostatin Analogues Containing Sugar Amino Acids
pp. 666
A Potent Non-Peptide Inhibitor of Anthrax Lethal Factor
pp. 668
Highly Potent Analogs of Human Parathyroid Hormone and Human Parathyroid Hormone-Related Protein
pp. 670
Glucagon-Like Peptide-1 Analogs with Significantly Improved in vivo Activity
pp. 672
Neuropeptide Y (NPY) Y1 Receptor Antagonists
pp. 674
Template-Directed Ligation of Peptides with Nucleobase Amino Acids
pp. 676
A General New Concept for the Development of Opioid Peptide Derived μ-, δ- and κ-Antagonists
pp. 679
Synthesis and Pharmacological Activity of Dmt-Tic Analogs with Highly Potent Agonist and Antagonist/Agonist Opioid Activity
pp. 681
A Novel Cyclic Opioid Peptide Antagonist Containing a Hydroxy Group in Place of the N-Terminal Amino Function
pp. 683
Modifications of the Tic Residue in TIPP-Peptides
pp. 685
Structure-Activity Relationships of Linear and Cyclic Nociceptin Analogs and Conformational Analysis by CD and NMR Spectroscopy
pp. 687
Design and Synthesis of Dynorphin A-(1–11) Analogs with C-Terminal Modifications and Evaluation of their Opioid Activity
pp. 689
C-Terminal Structure-Activity Relationships for the Novel Opioid Peptide JVA-901 (Venorphin)
pp. 691
Design and Synthesis of Bifunctional Peptides: Antagonists at CCKA/CCKB Receptors and Agonists at μ/δ Opioid Receptors
pp. 693
Role of the C-Terminal and Central Region of Gastrin for Recognition by the Human CCK2 Receptor
pp. 695
Structure and Peptide Binding Specificity of the SH3 and SH2 Domain from a Self-Regulated Protein Tyrosine Kinase — BTK
pp. 697
Pseudoprolines for Studying Bioactive cis-Prolyl Conformations
pp. 699
Design of Oxytocin Antagonists Which Are More Selective than Atosiban in Rat Bioassays and in Human Receptor Assays
pp. 701
Highly Selective Cyclic Peptides for Human Melanocortin-4 Receptor (MC-4 R): Design, Synthesis, Bioactive Conformation, and Pharmacological Evaluation as an Anti-Obesity Agent
pp. 704
SAR of Melanin-concentration Hormone (MCH), an Important Regulatory Hormone in Feeding Behavior
pp. 706
Structure-Activity Relationship Studies (SAR) of Melanocortin Agonists Central His-Phe-Arg-Trp Sequence
pp. 708
The Development of a Novel Highly Selective and Potent Agonist for Human Melanocortin 4 Receptor
pp. 710
Synthesis and NMR Characterization of Melanin-Concentrating Hormone
pp. 712
Synergism Between Agouti Protein Fragment 91–131 and Melanin Concentrating Hormone
pp. 714
Development of a Human Growth Hormone Peptide Analogue AOD9604 into an Anti-Obesity Drug
pp. 716
Rational Approach to Stable, Universal Somatostatin Analogues with Superior Therapeutic Potential
pp. 719
N-Methyl Scan of a sst1-Selective Somatostatin (SRIF) Analog
pp. 721
Exploring the “Double-Ring” Motif in Bradykinin Antagonists
pp. 723
Conformational Studies of Angiotensin II Cyclic Analogues
pp. 725
Identification of Key-Residues of Urotensin II, a Potent Mammalian Vasoconstrictor
pp. 727
Structure-Activity Studies on the Corticotropin Releasing Factor Antagonist Astressin, Minimal Sequence Necessary for Antagonistic Activity: Implications for a New Pharmacophoric Model
pp. 729
Solid-Phase Synthesis and Radiolabeling of a Bombesin Peptide Analog for Diagnostic Imaging of Tumors: A Preliminary Report
pp. 731
Investigation on the Structural Requirements for Binding Integrin αIIbβ3
pp. 733
Linear and Cyclic Peptides for Integrin αvβ6 Inhibition
pp. 735
The Synthesis of Collagen Peptides and Characterization of Their Inhibitory Effects on the Collagen Binding Activities of Integrins α1β1 and α2β1
pp. 737
Probing the Importance of the N-Terminal Helix of Parathyroid Hormone: Introduction of Cyclohexylalanine to Tether to the Membrane
pp. 739
Structure-Function Relationship Studies on Parathyroid Hormone (PTH) 1–34 Analogs Containing β-Amino Acid Residues in Positions 11, 12, and 13
pp. 742
Local Conformation Around Position 12 of the (1–34) Fragment of Parathyroid Hormone Probed by Substitution with Aib Residues
pp. 744
Positional Cyclization Scanning: A New Method to Evaluate the Bioactive Conformation of Glucagon
pp. 746
Age-Related Decreases of Calcitonin Gene-Related Peptide (CGRP)-Induced Hypotension in vivo and Vasorelaxant Responses in vitro in Rats
pp. 748
A Novel Series of Growth Hormone Secretagogues
pp. 750
Chimeric Mastoparans: Biological Probes and Designer Secretagogues
pp. 752
Design of Cyclic α-Defensin Dimers as Channel Forming BuildingBlocks
pp. 754
The Effect of Multiple Substitution of Aliphatic Amino Acids on the Structure, Function and Mode of Action of Lytic Peptides
pp. 756
Three-Dimensional Structure of Big Defensin, a Novel Antimicrobial Peptide Isolated from Horseshoe Crab
pp. 758
Selective Bioactivity of Synthetic Amphipathic Peptides Against Murine Macrophages Infected with Brucella abortus
pp. 760
Antibacterial Peptides Derived from the C-Terminal Domain of the Hemolytic Lectin, CEL-III
pp. 762
Low Molecular Weight Ψ[CH2NH] Pseudopeptides Yield Potent Antimicrobial Agents
pp. 764
Synthesis and Study of the Antimicrobial Action of Cecropin A-Melittin Hybrids with Aib Substitution
pp. 766
Structure-Function Relationship of Gramicidin-Alamethicin Hybrid Analogs
pp. 768
Biaryl-Bridged Lipopeptides from Streptomyces sp. TÜ 6075
pp. 770
Generation of Bioactive Peptides Derived from Caseins Using a Lactobacillus helveticus Strain
pp. 772
Bioactive Peptides Produced by a Strain of Lactobacillus plantarum: Characterization and Partial Purification
pp. 774
Stilboflavins, a Natural Peptaibol Library from the Mold Stilbella flavipes
pp. 776
Cyclic Analogues of the Insect Antimicrobial Peptides Drosocin and Apidaecin
pp. 778
Interaction of Antithrombin III-Binding Domain in Heparins with Novel Heparin Binding Peptides
pp. 780
Antithrombin III-Derived Novel Heparin Binding Peptides Have an Antagonistic Effect on Heparins
pp. 782
The Octapeptide (Fragment of Differentiation Factor HLDF) Exhibits Nuclease Activity and Induces Apoptosis
pp. 785
In vivo Proteolytic Hemoglobin Products as Tissue Growth Promoters
pp. 787
Synthesis and Pharmacological Activity of Superagonists of the ORL1 Receptor
pp. 789
Rational Designing of CXCR-4 Agonists and Antagonists: Synthesis of Novel Cyclam Derivatives of Stromal Cell-Derived Factor (SDF-1)
pp. 791
A Computational Study of Conformational Properties for N-Methylated Azapeptide Models
pp. 793
Structural Requirements of Non-Mammalian Vasodilatory Peptide Maxadilan, an Excellent Agonist of PACAP Type 1 Receptors
pp. 795
Effect of Deficiency of Cytochrome C Oxidase Assembly Peptide Cox17p on Mitochondrial Functions and Respiratory-Chain in Mice
pp. 797
Circadian Rhythm Pacemaker Neuropeptide “PDF” in Nocturnal Insect Cricket Gryllus bimaculatus: cDNA Cloning, mRNA Expression, and Nuclear Localization
pp. 799
Design and Synthesis of the Hydroxamic Acid Variants Antitumorigenic and Antimetastatic Hydroxamate Based Ac-PHSXX′-NH2 Sequences
pp. 801
Design, Synthesis and Evaluation of Growth Regulating SDF-1 Peptides on Breast Carcinoma Cells
pp. 803
Components of Tissue-Specific Peptide Pools as Negative Regulators of Cell Growth
pp. 805
HPLC Analysis, Modeling, and Biological Studies of Antiproliferative Heterocyclic Carboxamides
pp. 807
Macrophage Chemotactic Response to Elastin-Derived VGVAPG and VGVPG Permutations: A Structure-Activity Relationship and Receptor Binding Assay
pp. 811
Analysis and Evaluation of Rational Designed Calcium Binding Sites in CD2
pp. 814
Structural Basis for Selective Binding of Integrins to Extracellular Matrix
pp. 816
Regulation of the Promoter Binding Activity of a Bacterial Sigma Factor Explored Using Segmental Isotopic Labeling and NMR Spectroscopy
pp. 818
Chemically Engineering the Prion Protein Using Stepwise SPPS and Expressed Protein Ligation
pp. 820
Covalent and Non-Covalent Oligomerization of the Transmembrane α-Helix 4 from the Cystic Fibrosis Conductance Regulator
pp. 822
CtrΔe13, a Calcitonin Receptor Isoform Lacking 14 Amino Acids in Transmembrane Helix 7: Structure and Topology
pp. 824
Transmembrane Segment Peptides of the Ff Phage Major Coat Protein Form Parallel Homodimers
pp. 826
Refined 3D Model of hMC4R and Docking Study for hMC4R with α-Melanocyte Stimulating Hormone Analogue Ligands
pp. 828
Effect of Detergents on Intramolecular Helix-Helix Packing in a Membrane-Based Peptide Derived from CFTR
pp. 830
Primary Amphipathic Shuttle Peptides: Structural Requirements and Interactions with Model Membranes
pp. 832
Synthesis, Purification, and Analysis of the Transmembrane Domain of Phospholamban
pp. 834
Verification of a μ Opioid Receptor Model by Site-Directed Mutagenesis
pp. 836
Solid-Phase Synthesis and Chemical Ligation of Transmembrane Segments of Rhodopsin
pp. 838
Ion Gating and Selectivity in Gramicidin A
pp. 841
Docking of Transmembrane Helices Into Four Helix Bundles in the High Affinity IgE Receptor
pp. 843
Helical Net Plots and Surface Lipophilicity Mapping of Transmembrane Helices of Integral Membrane Proteins: Aids to 3D Structure Determination of Integral Membrane Proteins
pp. 845
Studies on the Involvement of a His Residue of mt1 GPCR TM Helix V in the Interaction with Melatonin
pp. 847
Biosynthesis and Biophysical Studies of Domains of sTE2P, a Yeast G Protein-Coupled Receptor
pp. 849
Transmembrane Segment Mimic Peptides Containing Peptoid Residues
pp. 851
Computational Chemistry and Opioidmimetics: Receptor-Ligand Interactions of Dmt-Tic Peptides
pp. 853
Conformational Model of Signal Transduction in the Transmembrane Region of the AT-1 Receptor
pp. 855
Role of the Water Medium in the Process of Signal Transmission from Peptides to Cellular Receptors
pp. 857
Structure-Based Design, Synthesis, and Surface Plasmon Resonance (SPR) Detection of Antagonists of the Grb2 SH2 Domain
pp. 859
Global Conformational Constraint in the Design of a Grb2 SH2 Domain Inhibitor
pp. 862
Local Conformational Constraint in the Design of a Grb2 SH2 Domain Inhibitor
pp. 864
Further Studies of the Signaling Mechanisms of the Antitumor Somatostatin Analogue TT-232
pp. 866
Generation of Cellulose Membrane-Bound Peptides with Free C-Termini: A Useful Approach for PDZ Binding Studies
pp. 868
A Focused Library Approach to PTP Inhibitor Discovery Predicated on the X-ray Structure of a PTPIB-Bound Lead Compound
pp. 870
Synthesis of the Ras-RBD Protein Pair
pp. 873
The Proline-Rich Antibacterial Peptide Family Inhibits Chaperone-Assisted Protein Folding
pp. 876
Probing the Binding Site of a Heptahelical Peptide Pheromone Receptor Using Photoaffinity Labelling, Site-Directed Mutagenesis and Spectroscopic Approaches
pp. 879
The Naturally Occurring Melanocortin Antagonist Agouti-Related Protein (AGRP) Possesses Similar and Distinct Interactions at the MC4 Receptor Compared with Melanocortin Agonist
pp. 881
Identification of Regions of the Epidermal Growth Factor Receptor Involved in Ligand Binding Specificity Using a High Affinity Form of the Ectodomain
pp. 884
Thrombin Receptor Aromatic Residues for Edge-to-Face CH/π Interaction with Ligand Phe-2-phenyl Group
pp. 886
Regions of G-Protein-Coupled Receptors Identified by Multiple Sequence Alignment
pp. 888
Tools for the Identification of Receptor Dimmers: Synthesis and Biological Evaluation of On-Resin Dimerized, Photosensitive Analogues of Angiotensin II
pp. 890
Minimization of Parathyroid Hormone Using Simultaneous Multiple Peptide Synthesis: Implications for Structure Based Drug Design
pp. 892
Structure-Activity Relationship Studies of New Cyclic MSH Analogues Using Cloned-Human Melanocortin Receptors Lead to Greater Selectivity and Inverse Agonists
pp. 894
Structure-Activity Relationships of Arodyn, a Novel Dynorphin A-(1–11) Analogue
pp. 896
Neurohypophyseal Receptors-Ligands: Where We Are After the Landmark Rhodopsin Structure Determination
pp. 898
Synthesis, Bioactivity and Receptor Binding of Fluorescent NBD Labeled Analogs of the Tridecapeptide Mating Pheromone of Saccharomyces cerevisiae
pp. 900
Molecular Model of the BNP-NPR-A Receptor Complex
pp. 902
Characterizing the Interactions Between Cholecystokinin and the G-Protein Coupled Receptors CCK1 and CCK2: An NMR-Based Study
pp. 905
Human Colon Cancers Recognize N-Carboxymethyl Gastrin by a Non-CCK1, Non-CCK2 Receptor
pp. 907
Functional Characterization of Two Drosophila melanogaster Type A Allatostatin Receptors Expressed in CHO Cells
pp. 909
Receptor-Bound Conformation of α-Peptide of Transducin (Gt) is not Stabilized by a “π-Cation” Interaction but by Constrained Lactam Bridges Between Residues 341 and 350
pp. 911
Solution and Membrane-Bound Conformational Properties of a Peptide from the First Extracellular Loop of the Angiotensin II AT1 Receptor
pp. 913
Synthesis of a Biotinylated Chemotactic Peptide Analog as a Probe for Formylpeptide-Receptor Interaction
pp. 915
Specific Activation of the Insulin Receptor by the Transmembrane Domain Peptides
pp. 917
Cyclopentapeptides as Rigidified Templates for Probing Interactions with the AT-1 Receptors
pp. 919
Receptor Binding Site of Arg-Lys Triple Repeat in Nociceptin Superagonist
pp. 921
Identification of Novel Ligands for Vasopressin V2 Receptor from Positional Scanning Libraries
pp. 923
Diversity Generation and Guest-Templated Self-Sorting in Dynamic Combinatorial Libraries
pp. 925
NMR Studies of the Interaction of α-Bungarotoxin with a Mimotope of the Nicotinic Acetylcholine Receptor
pp. 927
Selection of Antagonists of Fibroblast Growth Factor from a Phage-Display Peptide Library
pp. 931
Peptide Carrier for Efficient Drug Transport Into Living Cells
pp. 933
Design of Novel Cell Penetrating Peptides
pp. 935
Synthesis and Targeting with Novel Multi-Mannosylated Glycopeptide Modules
pp. 937
Liposaccharides: Utilisation for Peptide Delivery and for Enhancing Synthetic Peptide Immunogenicity
pp. 940
Down-Regulation of HIV-1 Long Terminal Repeat Controlled Viral Transcription by DNA-Binding, Arginine-Rich Fusion Proteins Derived from HIV-1 TAT for the Direct Delivery into the Nucleus
pp. 942
New Insights Into the Membrane Translocating Process of the Tat Peptide Used for Cellular Delivery of Various Biological Molecules
pp. 944
DUROS® Osmotic Implant for the Delivery of Peptides and Proteins
pp. 946
Utilization of ICAM-1 Peptide Conjugates for Drug Targeting to T-Cells
pp. 948
Regulation of Cadherin-Cadherin Interaction: Secondary Structure of the HAV and ADT Peptides Derived from Human E-Cadherin Sequence
pp. 950
Translocation of Various Arginine-Rich Peptides and the Potential of These Peptides as Carriers for Intracellular Protein Delivery
pp. 953
Reversible PEGylation: Thiolytic Regeneration of Active Protein from Its Polymer Conjugates
pp. 955
Lipoamino Acid and Liposaccharide Conjugated Peptides: Enhancement of Bioavailability
pp. 957
Regulation and Multiplicity of Peptide Transporters in Model Systems
pp. 959
A Novel Class of Cell Permeable “Karyophilic” Peptides: NLS-Mediated Nuclear Import of Dermaseptin Derived Peptides in Intact Cells
pp. 961
Characterization of Translocation Behavior of Arginine-Rich Membrane-Permeable Peptides
pp. 963
Structure and Activity of the N-Terminal Peptides of HIV-1 Glycoprotein 41 Types M (Major) and O (Outlier)
pp. 965
Specific Cleavage at Lys-147/Gly-148 in the Serine Protease Domain of Human Factor IXaβ by Plasmin: Effect on Catalytic Efficiency and Factor Villa Binding
pp. 967
Stability and Peptide Binding Specificity of BTK SH2 Domain: Molecular Basis for X-Linked Agammaglobulinemia
pp. 969
Designing Peptide Drugs/Ligands for Pathological States. A New Paradigm for Design of Bioactive Peptide Hormones and Neurotransmitters
pp. 971
Alternate Aggregation Pathways of Alzheimer β-Amyloid Peptides
pp. 973
Diabetes mellitus (DM) Causes Severe Impairment of Hypotensive Responses in vivo and Vasorelaxant Responses in vitro to the Neuropeptide CGRP
pp. 975
Triple-Helical Peptide Analysis of Collagenolytic Protease Activity
pp. 978
Design of More Potent, Radioiodinatable and Fluorescent Vasopressin Hypotensive Peptide Agonists
pp. 980
Antagonism of the Neurochemical Effect of Thyrotropin-Releasing Hormone by Its Peptide Analog
pp. 982
Synthesis of Selective Substrates for Syk PTK
pp. 984
Synthesis of Potent and Enzymatically Stable 4–18F-Benzoyl-NT(8–13) Analogs for Tumour Diagnosis Using PET
pp. 986
In vivo Imaging of Protease Activity and Drug Screening
pp. 988
Passive Repression of HIV-1 Long Terminal Repeat Enhancer Controlled Viral Transcription in HIV-1 Infected Cells by Cationic DNA-Binding Fusion Proteins
pp. 990
Passive Repression of HIV-1 Long Terminal Repeat Controlled Viral Transcription by Site-Directed Combinatorial Design of Artificial DNA-Binding Proteins Screened from Combinatorial Chemical Libraries
pp. 992
Fluorescent Biosensor for CrkII Phosphorylation by the Abl Tyrosine Kinase
pp. 994
Antibodies to Distinct Protein Epitopes from a Single Polyclonal Serum
pp. 996
Epitope Mapping of Anti-Type I Collagen Crosslinked N-Telopeptide Antibody with Synthetic Peptides
pp. 998
The Use of a Synthetic Biotinylated Peptide Probe for the Isolation of Adenomatous Polyposis Coli (APC) Tumor Suppressor Protein Complexes
pp. 1000
Folding and Peptide Binding of TPR Motifs from SGT
pp. 1002
CCT mRNA and CREB Phosphorylation Up Regulated by Peptide ZNC(C)PR in Rat Hippocampus
pp. 1004
A Combination of HER-2 Peptide Epitope Vaccines Mediate Superior Biological Effects
pp. 1006
Multivalent Vaccine Studies for HTLV-1 Associated Diseases
pp. 1008
Evaluation of HTLV-1 Cytotoxic T-Cell Epitopes in HLA-A2.1 Transgenic Mice
pp. 1010
New Branched Polypeptide Based Epitope-Conjugates: Synthesis and Immunrecognition
pp. 1012
Evaluation of Synergistic Interaction Between Cytokines and Peptide Epitope Vaccines in Protection Against HER-2 Expressing Lung Metastases
pp. 1014
Novel Classes of Neutrophil-Activating Peptides: Isolation and Their Physiological Significance
pp. 1016
Affinity of the HIV-1-Neutralizing Monoclonal Antibody 2F5 for gp41 ELDKWA Peptide Analogues
pp. 1018
A Discontinuous Antigenic Site Is Functionally Reproduced by Synthetic Peptide Constructions
pp. 1021
Four-Segment Tandem Ligation of Proteins with Unusual Branched Architecture
pp. 1023
Identification and Optimization of HIV-Specific CTL Antigens for Vaccine Design
pp. 1025
The Natural T-Helper Cell Epitope Repertoire is Unlikely to Contain Glycopeptides with Extended Carbohydrate Side-Chains
pp. 1027
Peptide Analogues of a Subdominant Epitope Expressed in EBV-Associated Tumors: Synthesis and Activity
pp. 1029
Synthetic Epitopes from Equine Infectious Anemia Virus (EIAV) Surface and Core Proteins
pp. 1031
B-Cell Linear Epitopes in the Conservative Regions of Hepatitis C Virus Envelope Glycoproteins
pp. 1033
Synthesis of a Covalently Reactive Antigen Analog Derived from a Conserved Sequence of HIV-1 gp120
pp. 1035
Isolation, cDNA Cloning, and Chemical Synthesis of Oryctes rhinoceros Defensin
pp. 1037
Deamidation within a γ-Gliadin-Derived Peptide Enhances Its Recognition by Serum Antibodies of CD Patients
pp. 1039
Identification of Conserved HIV-1-Derived Helper T Lymphocyte Epitopes Using Synthetic Peptides and High Throughput Binding Assays
pp. 1041
Determining the Fate of Glycopeptides During Antigen Processing in Antigen Presenting Cells
pp. 1043
Evaluation of Immune Response Elicited by Peptide Libraries Against Foot-and-Mouth Disease Virus
pp. 1045
Peptoid-Peptide Hybrids: Design, Synthesis and MHC Binding
pp. 1047
Synthetic Glycopeptide Models of MUC1 Core Protein
pp. 1049
Cathepsin D Produces the Potent Antimicrobial Peptide Parasin I from Histone H2A in Scaleless Fish Skin
pp. 1051
Characterization of Highly Stimulatory T Cell Ligands Identified Using Positional Scanning Libraries
pp. 1053
Proteomics Approach for Identifying Interacting Partners of a C-Terminal Functional Peptide Derived from the Tumor Suppressor, p21cip/waf1
pp. 1055
Cuvette-Based Biosensors as Micropreparative Affinity Surfaces
pp. 1057
A Comprehensive Database of Protein-Protein Interactions
pp. 1060
Cell Attachment and Neurite Outgrowth Activities of Laminin Peptide-Conjugated Chitosan Membrane
pp. 1063
Peptide-Amphiphile Induction of α-Helical Molecular Architecture and Interaction with Biomaterial Surfaces
pp. 1065
TOAC Peptides as Catalysts of Enantioselective Oxidations
pp. 1067
Synthesis of Arg-Gly-Asp-Ser Containing Oligopeptides and Evaluation of Their Cell-Attachment Activity
Similar content
3,293
Vulnerabilities and fisheries impacts: the uncertain future of manta and devil rays
Authors:
Donald Croll
,
William T. White
,
Bernie R Tershy
…
Thermal Interface Materials: Historical Perspective, Status, and Future Directions
Authors:
R. Prasher
Psychosocial job quality and mental health among young workers: a fixed-effects regression analysis using 13 waves of annual data
Authors:
Allison Milner
,
Lauren Krnjack
,
Anthony LaMontagne
See all similar
Cited by
1
Recent advances in covalent, site-specific protein immobilization
Authors:
Morten Meldal
,
Sanne Schoffelen
See all cited by